Pharmacology & ToxicologyToxicology LettersPeer-reviewed
Identification of ligands binding to MB327-PAM-1, a binding pocket relevant for resensitization of nAChRs
Jesko Kaiser, Christoph G. W. Gertzen, Tamara Bernauer…·Holger Gohlke
This paper identifies novel ligands binding to MB327-PAM-1, a binding site for resensitizing nAChRs, including cycloguanil, which shows higher affinity and functional efficacy.
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