BiochemistrybioRxivPreprint
A lipopeptidomimetic of transcriptional activation domains selectively disrupts Med25 PPIs
O. N. Pattelli, E. Martinez Valdivia, M. S. Beyersdorf…·A. K. Mapp
The paper develops a lipopeptidomimetic that selectively disrupts Med25 protein-protein interactions, showing improved affinity and selectivity for Med25 over other coactivators.
DOI 10.1101/2023.03.24.534168