BiochemistrybioRxivPreprint
Macrocyclization of an all-D linear peptide improves target affinity and imparts cellular activity: A novel stapled α-helical peptide modality
S. Kannan, P. G. A. Aronica, S. Ng…·A. Partridge
This paper combines macrocyclization and D-amino acid strategies to create an all-D helical peptide with improved target affinity and cellular activity.
DOI 10.1101/767673