Molecular insights into the atypical activation mechanism of GPR156 in maintaining auditory function
Xiangyu Ma, Li-Nan Chen, Menghui Liao, Liyan Zhang, Kun Xi, Jiamin Guo, Cangsong Shen, Dandan Shen, Pengjun Cai, Qingya Shen, Jieyu Qi, Huibing Zhang, Shao‐Kun Zang, Ying-Jun Dong, Luwei Miao, , Renjie Chai
This study reveals the constitutive activity and dimerization mechanism of GPR156, explaining its role in auditory function through cryo-EM structures and functional analysis.
bioRxiv · Mar 7, 2024 · PreprintMolecular Biology