Structural basis of Mycobacterium tuberculosis transcription and transcription inhibition
Wei Lin, Soma Mandal, David Degen, Yu Liu, Yon W. Ebright, Shengjian Li, Yu Feng, Yu Zhang, Sukhendu Mandal, Yi Jiang, Shuang Liu, Matthew Gigliotti, Meliza T. Talaue, Nancy D Connell, Kalyan Das, , Richard H. Ebright
This study reports crystal structures of Mycobacterium tuberculosis RNA polymerase with and without antituberculosis drugs, revealing a new class of inhibitors and their binding mechanisms.
Molecular Cell · Apr 1, 2017Peer-reviewedMolecular Biology