BiochemistryJournal of Medicinal ChemistryPeer-reviewed
Back-pocket optimization of 2-aminopyrimidine-based macrocycles leads to potent dual EPHA2/GAK kinase inhibitors with antiviral activity
Joshua Gerninghaus, Rezart Zhubi, Andreas Krämer…·Thomas Hanke
The paper optimizes a 2-aminopyrimidine-based macrocycle to create a dual EPHA2/GAK kinase inhibitor with antiviral activity against dengue virus.
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