Cancer BiologybioRxivPreprint
Rewiring DNA repair with PARP-based chemical inducers of proximity
Bryce da Camara, Eric M. Bilotta, Erin Broderick…·Michael A. Erb
This paper develops PCIP-1, a PARP-based chemical inducer of proximity that rewires DNA repair by recruiting BET proteins to PARP2, showing synthetic lethality in cancer cells with homologous recombination deficiencies.
3 citations