BioengineeringbioRxivPreprint
AI-Driven Efficient De Novo design of GLP-1RAs with Extended Half-Life and Enhanced Efficacy
Ting Wei, Xiaochen Cui, Jiahui Lin…·Haifeng Chen
This paper designs 10,000 de novo GLP-1RAs using AI, with 60 passing stability, efficacy, and diversity criteria, and two showing extended half-lives and superior efficacy in vivo.
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