MAPK Pathway Inhibition Reshapes Kinase Chemical Probe Reactivity Reflecting Cellular Activation States
Andrew F. Jarvis, Mohd Younis Bhat, Timothé Maujean, Ahlenne L. Abreu, Kaitlyn Toy, George M. Burslem, Donita C. Brady
This study uses ABPP to show how MAPK pathway inhibitors alter kinase residue reactivity, reflecting conformational changes and resistance mechanisms in melanoma cells.
ACS Bio & Med Chem Au · Jan 23, 2026Peer-reviewedCancer Biology