MicrobiologybioRxiv
Pharmacological and genetic activation of cAMP synthesis disrupts cholesterol utilization in Mycobacterium tuberculosis
K. M. Wilburn, C. R. Montague, B. Qin…·B. C. VanderVen
This paper identifies a small molecule agonist of Mtb adenylyl cyclase Rv1625c that inhibits cholesterol utilization and disrupts Mtb pathogenesis in mice.
DOI 10.1371/journal.ppat.1009862