Region-specific and dose-specific effects of chronic haloperidol exposure on Ro15-4513 GABA-A receptor binding sites in the rat brain
Alba Peris-Yague, Amanda Kiemes, Diana Cash…·Gemma Modinos
This study shows chronic haloperidol increases [3H]-Ro15-4513 binding in rat hippocampus and [3H]-flumazenil binding across brain regions, suggesting antipsychotics may affect GABAAR availability.