BiochemistryACS Medicinal Chemistry LettersPeer-reviewed
In vivo-Active Soluble Epoxide Hydrolase-targeting PROTACs with Improved Potency and Stability
Keita Nakane, Christophe H.P. Morisseau, Presley D. Dowker-Key…·Seiya Kitamura
This paper develops next-generation sEH-targeting PROTACs with improved potency and stability, showing effective degradation in mouse tissues.
6 citations