BiochemistryStructurePeer-reviewed
Discovery of Tankyrase scaffolding inhibitor specifically targeting the ARC4 peptide binding domain
Chiara Bosetti, Albert Galera‐Prat, Sven T. Sowa…·L. Lehtiö
The paper identifies a Tankyrase scaffolding inhibitor, S8 (ARCher-142), that selectively targets the ARC4 peptide binding domain with 8 µM potency.