MicrobiologyFEBS LettersPeer-reviewed
4-Nitrobenzoate inhibits 4-hydroxybenzoate polyprenyltransferase in malaria parasites and enhances atovaquone efficacy
Ignasi Bofill Verdaguer, Matheus Felipe Santos, Maurício Mazzine Filho…·Marcell Crispim
This study shows that 4-nitrobenzoate inhibits 4-HPT in malaria parasites, enhances atovaquone efficacy in vitro and in vivo, and identifies chemical requirements for this potentiation.