Cancer BiologybioRxivPreprint
Dyr726, a brain-penetrant inhibitor of PI3Kα, Type III receptor tyrosine kinases, and WNT signalling
Vasudha Tandon, Alessandra Fistrovich, Joaquina Nogales…·Sourav Banerjee
This paper designs and evaluates Dyr726, a brain-penetrant multi-kinase inhibitor that targets PI3Kα, receptor tyrosine kinases, and WNT signaling, showing efficacy in preclinical cancer models.
DOI 10.1101/2025.03.26.645490