BiochemistrybioRxivPreprint
Chemoproteomics identifies a pyrimidopyrimidine analogue as a tubulin-tyrosine ligase binder
Rubaba R Abanti, Eleftheria A. Georgiou, Dmytro Makarov…·Ioannis K. Kostakis
The paper identifies CEM198 as a TTL binder through chemoproteomics, showing it disrupts microtubule dynamics via dual mechanisms in different cell lines.
DOI 10.64898/2026.08.06.743276