BiochemistryBioconjugate ChemistryPeer-reviewed
NanoBRET Tracer Development for Class I Bromodomain Target Engagement in Live Cells
Molly Sneddon, Chi-Ming Tsou, Xiang Fu…·William C. K. Pomerantz
The paper develops a NanoBRET tracer, MS-1, to assess functional activity of class I bromodomain inhibitors in live cells, showing broad applicability across BPTF, PCAF, GCN5, and CECR2.
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