BiophysicsbioRxivPreprint
Molecular insights into inhibitor action on a key bacterial metabolic enzyme Cystathionine β-Synthase
Sainath Polepalli, Anupam Roy, Bapan Mondal…·Somnath Dutta
This paper investigates the molecular mechanism of aminooxyacetic acid (AOAA) inhibition of MtbCBS, a key bacterial enzyme, using cryo-EM and computational methods, revealing critical residues and structural factors for irreversible inhibition.
DOI 10.1101/2025.07.03.662948