Identification of novel human 15-lipoxygenase-2 (h15-LOX-2) inhibitors using a virtual screening approach
Lucas Gasparello Viviani, Thais Satie Iijima, Erika Piccirillo, Leandro de Rezende, Thiago Gerônimo Pires Alegria, Luís Eduardo Soares Netto, Antônia Tavares do Amaral, Sayuri Miyamoto
This study identifies six novel h15-LOX-2 inhibitors using virtual screening from a curated ZINC database, with two showing micromolar potency and a mixed-type inhibition mechanism.
Journal of Medicinal Chemistry · Dec 19, 2024Peer-reviewedBiochemistry