Integrative in silico and experimental identification of non-covalent UBE2N inhibitors enhancing PARP inhibitor sensitivity
Côme Ghadi, Shafi Ullah Khan, Léonie Ibazizene, Florian Schwalen, Charline Kieffer, Peggy Suzanne, Julie Jaouen, Hassiba Bouafia, Xavier Thuru, Marie Cornu, Cédric Lecoutey, Matthieu Meryet‐Figuière, Anne Sophie Voisin‐Chiret, Louis‐Bastien Weiswald, Jana Sopková‐de Oliveira Santos
The paper identifies two non-covalent UBE2N inhibitors, CERMN-2 and CERMN-16, which enhance PARP inhibitor sensitivity in ovarian cancer cells.
European Journal of Medicinal Chemistry Reports · Jul 30, 2026Peer-reviewedCancer Biology