First-in-class -PET radiotracers for GPR39: A platform for noninvasive target engagement imaging in vivo
B. Bhoopal, R. W. Fitzgerald, K. Gollapelli, M. Miller, N. Damuka, C. Baity, P. Roy, P. Myburgh, D. Zhou, P. Jadiya, R. Cerevera-Juanes, K. K. Solingapuram Sai
This paper introduces [18F]GPR39 2.1, a PET radiotracer for noninvasive imaging of GPR39, showing high specificity and sensitivity in vivo.
bioRxiv · Nov 9, 2026 · PreprintNeuroscience