Cell BiologybioRxiv
Unprotected Peptide Macrocyclization and Stapling via A Fluorine-Thiol Displacement Reaction
M. S. Islam, S. L. Junod, S. Zhang…·R. E. Wang
This paper introduces a new peptide stapling method using fluorine-thiol displacement reaction, showing improved stability, affinity, and cell permeability compared to traditional methods.
DOI 10.1038/s41467-022-27995-5