Second-Generation Cap Analogue Prodrugs for Targeting Aberrant Eukaryotic Translation Initiation Factor 4E (eIF4E) Activity in Drug-Resistant Melanoma
Emilio L. Cárdenas, Rachel L. O’Rourke, Arya Menon, Gabriela Vega-Hernández, Jennifer L. Meagher, Jeanne A. Stuckey, Amanda L. Garner
This study develops second-generation cap analogue inhibitors to target eIF4E-mediated cap-dependent translation in drug-resistant melanoma cells.
bioRxiv · Sep 25, 2024 · PreprintCancer Biology