Cancer BiologyMolecular & Cellular ProteomicsPeer-reviewed
CellEKT: A robust chemical proteomics workflow to profile cellular target engagement of kinase inhibitors
Joel Rüegger, Berend Gagestein, Antonius P. A. Janssen…·Mario van der Stelt
CellEKT profiles cellular target engagement of kinase inhibitors using chemical proteomics to determine IC50 values across over 300 kinases and validate results with phosphoproteomics and NanoBRET.
10 citations