Dizocilpine derivatives with neuroprotective effect lacking the psychomimetic side effects
Jan Konecny, Anna Misiachna, Markéta Chvojková, Lenka Kletečková, Marharyta Kolcheva, Martin Novák, Lukáš Prchal, Marek Ladislav, Katarína Hemelíková, Jakub Netolický, Martina Hrabinová, Tereza Kobrlová, Jana Žďárová Karasová, Jaroslav Pejchal, Pavla Jendelová, , Martin Hořák
This study develops novel NMDA receptor antagonists with neuroprotective effects and reduced psychomimetic side effects through structural modifications of MK-801.
bioRxiv · Jun 17, 2024 · PreprintNeuroscience