NeurosciencebioRxivPreprint
A functionally conserved mechanism of modulation via a vestibule site in pentameric ligand-gated ion channels
Marijke Brams, Cédric Govaerts, Kumiko Kambara…·Chris Ulens
The paper identifies a conserved vestibule binding site in pLGICs and shows nanobodies can act as allosteric modulators, expanding drug design possibilities.
DOI 10.1101/770719