Pharmacology & ToxicologybioRxivPreprint
Identification of Direct-acting nsP2 Helicase Inhibitors with Anti-alphaviral Activity
M. Bose, John D. Sears, Kacey Marie Talbot…·Timothy Mark Willson
This paper identifies and optimizes oxaspiropiperidine inhibitors targeting nsP2hel, showing nanomolar antiviral activity against multiple alphaviruses.