Structural, biophysical, and virological mechanistic characterization of HIV-1 capsid-targeting antivirals
Karen A. Kirby, William M. McFadden, Lin Wang, Haijuan Du, Huanchun Zhang, Andres Emanuelli Castaner, Zachary C. Lorson, Arvin Nafisi, Anastasia Selyutina, Charlotte Luchsinger, Atsuko Hachiya, Maria E. Cilento, Alexa A. Snyder, S Ravichandran, Xinyong Cai, , Stefan G. Sarafianos
The paper characterizes structural, biophysical, and virological properties of HIV-1 capsid-targeting antivirals, showing improved potency and stability through chemical modifications of PF74.
bioRxiv · Mar 25, 2026 · PreprintBiochemistry